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Abstract #2990

Imaging Extracellular Lactate with Lanthanide-PCTA-based PARACEST Agents

Remy Chiaffarelli1,2, Paul Jurek3, Pedro Cruz4, Max Zimmermann1,2, Carlos Geraldes4, Garry Kiefer3, and André Ferreira Martins1,2
1Werner Siemens Imaging Center, Department of Preclinical Imaging and Radiopharmacy, University Hospital Tuebingen, Tuebingen, Germany, 2Cluster of Excellence iFIT (EXC 2180) “Image-Guided and Functionally Instructed Tumor Therapies”, University of Tuebingen, Tuebingen, Germany, 3Macrocyclics, Inc., Plano, TX, United States, 4Coimbra Chemistry Center - Institute of Molecular Sciences (CQC-IMS), University of Coimbra, Coimbra, Portugal

Synopsis

Keywords: CEST & MT, CEST & MT, PARACEST, MetabolismLactate accumulation in the tumor microenvironment is a hallmark of cancer aggressiveness. Here, we report a method to image extracellular lactate using shiftCEST MRI and Yb- and EuPCTA Shift Reagents (SRs). In the presence of lactate, the SRs shift the lactate OH-CEST signal away from the water signal by ~14 ppm (EuPCTA) and ~95 ppm (YbPCTA), allowing for quantitative detection of extracellular lactate produced by cancer cells. In vivo studies confirmed the detection and fast renal elimination of the lactate*YbPCTA into the bladder by shiftCEST MRI. Overall, these results provide new insights into developing innovative non-invasive metabolic MRI.

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